| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 1 |
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| Ligand | BDBM42423 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose response cell-based screening assay for antagonists of neuropeptide Y receptor Y1 (NPY-Y1) |
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| IC50 | 6687±n/a nM |
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| Citation |  PubChem, PC Dose response cell-based screening assay for antagonists of neuropeptide Y receptor Y1 (NPY-Y1) PubChem Bioassay(2008)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Neuropeptide Y receptor type 1 |
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| Name: | Neuropeptide Y receptor type 1 |
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| Synonyms: | NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44399.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | NPY-Y1 NPY1R HUMAN::P25929 |
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| Residue: | 384 |
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| Sequence: | MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI
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| BDBM42423 |
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| n/a |
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| Name | BDBM42423 |
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| Synonyms: | MLS000519450 | SMR000129869 | [1-(4-chlorobenzyl)indol-3-yl]-(2-furyl)methanone | [1-[(4-chlorophenyl)methyl]-3-indolyl]-(2-furanyl)methanone | [1-[(4-chlorophenyl)methyl]indol-3-yl]-(furan-2-yl)methanone | cid_955150 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H14ClNO2 |
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| Mol. Mass. | 335.784 |
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| SMILES | Clc1ccc(Cn2cc(C(=O)c3ccco3)c3ccccc23)cc1 |
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| Structure | 
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