| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Neuropeptide Y receptor type 1 |
|---|
| Ligand | BDBM41946 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism |
|---|
| IC50 | 5388±n/a nM |
|---|
| Citation |  PubChem, PC Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism PubChem Bioassay(2008)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Neuropeptide Y receptor type 1 |
|---|
| Name: | Neuropeptide Y receptor type 1 |
|---|
| Synonyms: | NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 44399.07 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | NPY-Y1 NPY1R HUMAN::P25929 |
|---|
| Residue: | 384 |
|---|
| Sequence: | MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLA
LIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQ
CVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMT
DEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKR
RNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNL
LFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVS
KTSLKQASPVAFKKINNNDDNEKI
|
|
|
|---|
| BDBM41946 |
|---|
| n/a |
|---|
| Name | BDBM41946 |
|---|
| Synonyms: | 3-(2-bromanyl-6-chloranyl-4-methyl-phenoxy)-N-(phenylmethyl)propan-1-amine;ethanedioic acid | 3-(2-bromo-6-chloro-4-methylphenoxy)-N-(phenylmethyl)-1-propanamine;oxalic acid | MLS000576317 | N-benzyl-3-(2-bromo-6-chloro-4-methylphenoxy)-1-propanamine oxalate | N-benzyl-3-(2-bromo-6-chloro-4-methylphenoxy)propan-1-amine;oxalic acid | SMR000197957 | benzyl-[3-(2-bromo-6-chloro-4-methyl-phenoxy)propyl]amine;oxalic acid | cid_2933964 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H19BrClNO |
|---|
| Mol. Mass. | 368.696 |
|---|
| SMILES | Cc1cc(Cl)c(OCCCNCc2ccccc2)c(Br)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
