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TargetSignal transducer and activator of transcription 3 [702-738,740-752]
LigandBDBM46337
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based assay to measure STAT3 inhibition
IC50 5020±n/a nM
Citation PubChem, PC Dose response cell-based assay to measure STAT3 inhibition PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Signal transducer and activator of transcription 3 [702-738,740-752]
Name:Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:APRF | STAT3 | STAT3_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:5263.93
Organism:Homo sapiens (Human)
Description:gi_13272532
Residue:50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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BDBM46337
n/a
NameBDBM46337
Synonyms:1-[5-(4-Chloro-benzylsulfanyl)-[1,3,4]oxadiazol-2-ylmethyl]-1H-benzoimidazole | 2-(1-benzimidazolylmethyl)-5-[(4-chlorophenyl)methylthio]-1,3,4-oxadiazole | 2-(benzimidazol-1-ylmethyl)-5-[(4-chlorobenzyl)thio]-1,3,4-oxadiazole | 2-(benzimidazol-1-ylmethyl)-5-[(4-chlorophenyl)methylsulfanyl]-1,3,4-oxadiazole | MLS000030897 | SMR000001594 | cid_646906
TypeSmall organic molecule
Emp. Form.C17H13ClN4OS
Mol. Mass.356.829
SMILESClc1ccc(CSc2nnc(Cn3cnc4ccccc34)o2)cc1
Structure
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