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TargetSignal transducer and activator of transcription 3 [702-738,740-752]
LigandBDBM46338
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based assay to measure STAT3 inhibition
IC50 6728±n/a nM
Citation PubChem, PC Dose response cell-based assay to measure STAT3 inhibition PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Signal transducer and activator of transcription 3 [702-738,740-752]
Name:Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:APRF | STAT3 | STAT3_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:5263.93
Organism:Homo sapiens (Human)
Description:gi_13272532
Residue:50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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BDBM46338
n/a
NameBDBM46338
Synonyms:2-[1-(2,3-Dihydro-benzo[1,4]dioxine-6-sulfonyl)-piperidin-4-yl]-benzothiazole | 2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-piperidinyl]-1,3-benzothiazole | 2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)-4-piperidyl]-1,3-benzothiazole | 2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)piperidin-4-yl]-1,3-benzothiazole | MLS000073837 | SMR000007058 | cid_651062
TypeSmall organic molecule
Emp. Form.C20H20N2O4S2
Mol. Mass.416.514
SMILESO=S(=O)(N1CCC(CC1)c1nc2ccccc2s1)c1ccc2OCCOc2c1
Structure
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