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TargetSignal transducer and activator of transcription 3 [702-738,740-752]
LigandBDBM46396
Substrate/Competitorn/a
Meas. Tech.Dose response cell-based assay to measure STAT3 inhibition
IC50 3700±n/a nM
Citation PubChem, PC Dose response cell-based assay to measure STAT3 inhibition PubChem Bioassay(2008)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Signal transducer and activator of transcription 3 [702-738,740-752]
Name:Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:APRF | STAT3 | STAT3_HUMAN
Type:Enzyme Catalytic Domain
Mol. Mass.:5263.93
Organism:Homo sapiens (Human)
Description:gi_13272532
Residue:50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
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BDBM46396
n/a
NameBDBM46396
Synonyms:MLS000589892 | N-(3-Hydroxy-phenyl)-N'-pyridin-2-yl-oxalamide | N-(3-hydroxyphenyl)-N'-(2-pyridinyl)oxamide | N-(3-hydroxyphenyl)-N'-(2-pyridyl)oxamide | N-(3-hydroxyphenyl)-N'-pyridin-2-yl-ethanediamide | N-(3-hydroxyphenyl)-N'-pyridin-2-yloxamide | SMR000217071 | cid_1898255
TypeSmall organic molecule
Emp. Form.C13H11N3O3
Mol. Mass.257.2447
SMILESOc1cccc(NC(=O)C(=O)Nc2ccccn2)c1
Structure
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