| Reaction Details |
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 | Report a problem with these data |
| Target | D(1A) dopamine receptor |
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| Ligand | BDBM48909 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Allosteric Modulators of D1 Receptors: Dose-dependent Assay |
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| EC50 | 0.0101±n/a nM |
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| Citation |  PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Assay PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| D(1A) dopamine receptor |
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| Name: | D(1A) dopamine receptor |
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| Synonyms: | DA D1 receptor | DOPAMINE D1 | DRD1 | DRD1_HUMAN | Dopamine D1 receptor | Dopamine D1 receptor (D1R) | Dopamine D1A |
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| Type: | Enzyme |
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| Mol. Mass.: | 49303.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21728 |
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| Residue: | 446 |
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| Sequence: | MRTLNTSAMDGTGLVVERDFSVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTN
FFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVD
RYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNATSLA
ETIDNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKN
CQTTTGNGKPVECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCGS
GETQPFCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPATNNAIET
VSINNNGAAMFSSHHEPRGSISKECNLVYLIPHAVGSSEDLKKEEAAGIARPLEKLSPAL
SVILDYDTDVSLEKIQPITQNGQHPT
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| BDBM48909 |
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| n/a |
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| Name | BDBM48909 |
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| Synonyms: | 2-[5-(4-Fluoro-phenyl)-thiazolo[2,3-c][1,2,4]triazol-3-ylsulfanyl]-N-furan-2-ylmethyl-acetamide | 2-[[5-(4-fluorophenyl)-3-thiazolo[2,3-c][1,2,4]triazolyl]thio]-N-(2-furanylmethyl)acetamide | 2-[[5-(4-fluorophenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]sulfanyl]-N-(furan-2-ylmethyl)acetamide | 2-[[5-(4-fluorophenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl]sulfanyl]-N-(furan-2-ylmethyl)ethanamide | 2-[[5-(4-fluorophenyl)thiazolo[2,3-c][1,2,4]triazol-3-yl]thio]-N-(2-furfuryl)acetamide | MLS000068421 | SMR000007125 | cid_649740 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H13FN4O2S2 |
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| Mol. Mass. | 388.439 |
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| SMILES | Fc1ccc(cc1)-c1csc2nnc(SCC(=O)NCc3ccco3)n12 |
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| Structure | 
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