Ki Summary

Reaction Details

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Target

Dual specificity protein phosphatase 3

Ligand

BDBM50703

Substrate/Competitor

n/a

Meas. Tech.

uHTS absorbance assay for the identification of compounds that inhibit VHR1.

IC50

10400±n/a nM

Citation

PubChem, PC uHTS absorbance assay for the identification of compounds that inhibit VHR1. PubChem Bioassay(2009)[AID]

More Info.:

Get all data from this article, Solution Info, Assay Method

Dual specificity protein phosphatase 3

Name:

Dual specificity protein phosphatase 3

Synonyms:

Type:

Hydrolase

Mol. Mass.:

20480.58

Organism:

Homo sapiens (Human)

Description:

n/a

Residue:

185

Sequence:

MSGSFELSVQDLNDLLSDGSGCYSLPSQPCNEVTPRIYVGNASVAQDIPKLQKLGITHVL
NAAEGRSFMHVNTNANFYKDSGITYLGIKANDTQEFNLSAYFERAADFIDQALAQKNGRV
LVHCREGYSRSPTLVIAYLMMRQKMDVKSALSIVRQNREIGPNDGFLAQLCQLNDRLAKE
GKLKP

BDBM50703

n/a

Name

BDBM50703

Synonyms:

3-[1-(3,4-Dihydroxy-phenyl)-meth-(E)-ylidene]-4-imino-7-methanesulfonyl-3,4-dihydro-9-thia-1,4a-diaza -fluoren-2-one | 4-amino-3-[(Z)-(3-hydroxy-4-keto-cyclohexa-2,5-dien-1-ylidene)methyl]-8-mesyl-pyrimido[2,1-b][1,3]benzothiazol-2-one | 4-amino-3-[(Z)-(3-hydroxy-4-oxo-1-cyclohexa-2,5-dienylidene)methyl]-8-methylsulfonyl-2-pyrimido[2,1-b][1,3]benzothiazolone | 4-amino-3-[(Z)-(3-hydroxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-8-methylsulfonylpyrimido[2,1-b][1,3]benzothiazol-2-one | 4-azanyl-8-methylsulfonyl-3-[(Z)-(3-oxidanyl-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)methyl]pyrimido[2,1-b][1,3]benzothiazol-2-one | MLS000779134 | SMR000415838 | cid_16682713

Type

Small organic molecule

Emp. Form.

C18H13N3O5S2

Mol. Mass.

415.443

SMILES

CS(=O)(=O)c1ccc2c(c1)sc1nc(=O)c(\C=C3\C=CC(=O)C(O)=C3)c(N)n21 |c:19,24|

Structure