| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptides B/W receptor type 1 |
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| Ligand | BDBM62144 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence-based dose response cell-based high throughput screening assay to identify antagonists of the G-protein coupled receptor 7 (GPR7). |
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| IC50 | 23855±n/a nM |
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| Citation |  PubChem, PC Fluorescence-based dose response cell-based high throughput screening assay to identify antagonists of the G-protein coupled receptor 7 (GPR7). PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Neuropeptides B/W receptor type 1 |
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| Name: | Neuropeptides B/W receptor type 1 |
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| Synonyms: | GPR7 | NPBW1_HUMAN | NPBWR1 | neuropeptides B/W receptor 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36111.82 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_119607128 |
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| Residue: | 328 |
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| Sequence: | MDNASFSEPWPANASGPDPALSCSNASTLAPLPAPLAVAVPVVYAVICAVGLAGNSAVLY
VLLRAPRMKTVTNLFILNLAIADELFTLVLPINIADFLLRQWPFGELMCKLIVAIDQYNT
FSSLYFLTVMSADRYLVVLATAESRRVAGRTYSAARAVSLAVWGIVTLVVLPFAVFARLD
DEQGRRQCVLVFPQPEAFWWRASRLYTLVLGFAIPVSTICVLYTTLLCRLHAMRLDSHAK
ALERAKKRVTFLVVAILAVCLLCWTPYHLSTVVALTTDLPQTPLVIAISYFITSLSYANS
CLNPFLYAFLDASFRRNLRQLITCRAAA
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| BDBM62144 |
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| n/a |
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| Name | BDBM62144 |
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| Synonyms: | (4-ethyl-1-piperazinyl)-[4-[(4-methylphenyl)methyl]-2,3-dihydro-1,4-benzothiazin-6-yl]methanone | (4-ethylpiperazin-1-yl)-[4-[(4-methylphenyl)methyl]-2,3-dihydro-1,4-benzothiazin-6-yl]methanone | (4-ethylpiperazino)-[4-(4-methylbenzyl)-2,3-dihydro-1,4-benzothiazin-6-yl]methanone | MLS000925100 | SMR000624010 | cid_6622858 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H29N3OS |
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| Mol. Mass. | 395.561 |
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| SMILES | CCN1CCN(CC1)C(=O)c1ccc2SCCN(Cc3ccc(C)cc3)c2c1 |
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| Structure | 
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