| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM64861 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1) |
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| IC50 | 8637±n/a nM |
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| Citation |  PubChem, PC Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1) PubChem Bioassay(2010)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44789.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35372 |
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| Residue: | 400 |
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| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM64861 |
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| n/a |
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| Name | BDBM64861 |
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| Synonyms: | 5-(2,4-dichlorobenzyl)-2-(2-pyridinyl)-4,6-pyrimidinediamine | 5-[(2,4-dichlorophenyl)methyl]-2-(2-pyridinyl)pyrimidine-4,6-diamine | 5-[(2,4-dichlorophenyl)methyl]-2-pyridin-2-yl-pyrimidine-4,6-diamine | 5-[(2,4-dichlorophenyl)methyl]-2-pyridin-2-ylpyrimidine-4,6-diamine | MLS000691892 | SMR000333929 | [6-amino-5-(2,4-dichlorobenzyl)-2-(2-pyridyl)pyrimidin-4-yl]amine | cid_3379829 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H13Cl2N5 |
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| Mol. Mass. | 346.214 |
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| SMILES | Nc1nc(nc(N)c1Cc1ccc(Cl)cc1Cl)-c1ccccn1 |
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| Structure | 
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