| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Photoreceptor-specific nuclear receptor |
|---|
| Ligand | BDBM37784 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3) |
|---|
| IC50 | >39841±n/a nM |
|---|
| Citation |  PubChem, PC TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3) PubChem Bioassay(2010)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Photoreceptor-specific nuclear receptor |
|---|
| Name: | Photoreceptor-specific nuclear receptor |
|---|
| Synonyms: | NR2E3 | NR2E3_HUMAN | PNR | RNR | photoreceptor-specific nuclear receptor |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 44699.83 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | ChEMBL_401901 |
|---|
| Residue: | 410 |
|---|
| Sequence: | METRPTALMSSTVAAAAPAAGAASRKESPGRWGLGEDPTGVSPSLQCRVCGDSSSGKHYG
IYACNGCSGFFKRSVRRRLIYRCQVGAGMCPVDKAHRNQCQACRLKKCLQAGMNQDAVQN
ERQPRSTAQVHLDSMESNTESRPESLVAPPAPAGRSPRGPTPMSAARALGHHFMASLITA
ETCAKLEPEDADENIDVTSNDPEFPSSPYSSSSPCGLDSIHETSARLLFMAVKWAKNLPV
FSSLPFRDQVILLEEAWSELFLLGAIQWSLPLDSCPLLAPPEASAAGGAQGRLTLASMET
RVLQETISRFRALAVDPTEFACMKALVLFKPETRGLKDPEHVEALQDQSQVMLSQHSKAH
HPSQPVRFGKLLLLLPSLRFITAERIELLFFRKTIGNTPMEKLLCDMFKN
|
|
|
|---|
| BDBM37784 |
|---|
| n/a |
|---|
| Name | BDBM37784 |
|---|
| Synonyms: | 1-(2-furanylmethyl)-4-hydroxy-3-[(7-methoxy-2-benzofuranyl)-oxomethyl]-2-(3-pyridinyl)-2H-pyrrol-5-one | 1-(2-furfuryl)-3-hydroxy-4-(7-methoxybenzofuran-2-carbonyl)-5-(3-pyridyl)-3-pyrrolin-2-one | 1-(2-furylmethyl)-3-hydroxy-4-[(7-methoxy-1-benzofuran-2-yl)carbonyl]-5-(3-pyridinyl)-1,5-dihydro-2H-pyrrol-2-one | 1-(furan-2-ylmethyl)-3-[(7-methoxy-1-benzofuran-2-yl)carbonyl]-4-oxidanyl-2-pyridin-3-yl-2H-pyrrol-5-one | 1-(furan-2-ylmethyl)-4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-pyridin-3-yl-2H-pyrrol-5-one | MLS000097076 | SMR000075743 | cid_2951279 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C24H18N2O6 |
|---|
| Mol. Mass. | 430.4095 |
|---|
| SMILES | COc1cccc2cc(oc12)C(=O)C1C(N(Cc2ccco2)C(=O)C1=O)c1cccnc1 |
|---|
| Structure | 
|
|---|
Search and Browse
