Reaction Details |
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Target | Sentrin-specific protease 8 |
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Ligand | BDBM76363 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay |
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IC50 | 86800±n/a nM |
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Citation | PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID] |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Sentrin-specific protease 8 |
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Name: | Sentrin-specific protease 8 |
Synonyms: | DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8 |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 24104.52 |
Organism: | Homo sapiens (Human) |
Description: | gi_262118306 |
Residue: | 212 |
Sequence: | MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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BDBM76363 |
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n/a |
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Name | BDBM76363 |
Synonyms: | 4-(4-fluorophenyl)-N-phenyl-3,6-dihydro-1(2H)-pyridinecarboxamide | 4-(4-fluorophenyl)-N-phenyl-3,6-dihydro-2H-pyridine-1-carboxamide | MLS000100266 | SMR000082286 | cid_2980777 |
Type | Small organic molecule |
Emp. Form. | C18H17FN2O |
Mol. Mass. | 296.3388 |
SMILES | Fc1ccc(cc1)C1=CCN(CC1)C(=O)Nc1ccccc1 |t:8| |
Structure |
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