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TargetSentrin-specific protease 8
LigandBDBM69620
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay
IC50 5940±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sentrin-specific protease 8
Name:Sentrin-specific protease 8
Synonyms:DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8
Type:Enzyme Catalytic Domain
Mol. Mass.:24104.52
Organism:Homo sapiens (Human)
Description:gi_262118306
Residue:212
Sequence:
MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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  Blast E-value cutoff:
BDBM69620
n/a
NameBDBM69620
Synonyms:(4-bromophenyl)(5-hydroxy-1-benzofuran-3-yl)methanone | (4-bromophenyl)-(5-hydroxy-1-benzofuran-3-yl)methanone | (4-bromophenyl)-(5-hydroxy-3-benzofuranyl)methanone | (4-bromophenyl)-(5-hydroxybenzofuran-3-yl)methanone | (4-bromophenyl)-(5-oxidanyl-1-benzofuran-3-yl)methanone | MLS001178337 | SMR000476405 | cid_900927
TypeSmall organic molecule
Emp. Form.C15H9BrO3
Mol. Mass.317.134
SMILESOc1ccc2occ(C(=O)c3ccc(Br)cc3)c2c1
Structure
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