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TargetSentrin-specific protease 8
LigandBDBM76785
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay
IC50>100000±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Sentrin-specific protease 8
Name:Sentrin-specific protease 8
Synonyms:DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8
Type:Enzyme Catalytic Domain
Mol. Mass.:24104.52
Organism:Homo sapiens (Human)
Description:gi_262118306
Residue:212
Sequence:
MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQ
FIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDS
HSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFR
QQTESLLQLLTPAYITKKRGEWKDLITTLAKK
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  Blast E-value cutoff:
BDBM76785
n/a
NameBDBM76785
Synonyms:3-(3,5-dimethoxyphenyl)-2-benzopyran-1-one | 3-(3,5-dimethoxyphenyl)isochromen-1-one | 3-(3,5-dimethoxyphenyl)isocoumarin | MLS001360842 | SMR001216324 | cid_25058224
TypeSmall organic molecule
Emp. Form.C17H14O4
Mol. Mass.282.2907
SMILESCOc1cc(OC)cc(c1)-c1cc2ccccc2c(=O)o1
Structure
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