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TargetMitochondrial import inner membrane translocase subunit TIM10
LigandBDBM78181
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS small molecule inhibitors of tim10-1 yeast via a luminescent assay
IC50 6400±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS small molecule inhibitors of tim10-1 yeast via a luminescent assay PubChem Bioassay(2010)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Mitochondrial import inner membrane translocase subunit TIM10
Name:Mitochondrial import inner membrane translocase subunit TIM10
Synonyms:MRS11 | TIM10 | TIM10_YEAST | TPA: Essential protein of the mitochondrial intermembrane space | TPA: Essential protein of the mitochondrial intermembrane space, forms a complex with Tim9p (TIM10 complex) that delivers hydrophobic proteins to the TIM22 complex for insertion into the inner ...
Type:Enzyme Catalytic Domain
Mol. Mass.:10303.50
Organism:Saccharomyces cerevisiae S288c
Description:gi_285809906
Residue:93
Sequence:
MSFLGFGGGQPQLSSQQKIQAAEAELDLVTDMFNKLVNNCYKKCINTSYSEGELNKNESS
CLDRCVAKYFETNVQVGENMQKMGQSFNAAGKF
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BDBM78181
n/a
NameBDBM78181
Synonyms:(E)-3-(3-Benzotriazol-1-ylmethyl-4-methoxy-phenyl)-1-phenyl-propenone | (E)-3-[3-(1-benzotriazolylmethyl)-4-methoxyphenyl]-1-phenyl-2-propen-1-one | (E)-3-[3-(benzotriazol-1-ylmethyl)-4-methoxy-phenyl]-1-phenyl-prop-2-en-1-one | (E)-3-[3-(benzotriazol-1-ylmethyl)-4-methoxyphenyl]-1-phenylprop-2-en-1-one | MLS000589828 | SMR000217110 | cid_6184004
TypeSmall organic molecule
Emp. Form.C23H19N3O2
Mol. Mass.369.4159
SMILESCOc1ccc(\C=C\C(=O)c2ccccc2)cc1Cn1nnc2ccccc12
Structure
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