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TargetUbiquitin-conjugating enzyme E2 N
LigandBDBM43873
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay
IC50>20000±0 nM
Citation PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay(2011)[AID]
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Ubiquitin-conjugating enzyme E2 N
Name:Ubiquitin-conjugating enzyme E2 N
Synonyms:BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N
Type:PROTEIN
Mol. Mass.:17137.61
Organism:Homo sapiens (Human)
Description:EBI_101440
Residue:152
Sequence:
MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
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  Blast E-value cutoff:
BDBM43873
n/a
NameBDBM43873
Synonyms:1-[(Z)-[1-[(4-fluorophenyl)methyl]-2-oxidanylidene-indol-3-ylidene]amino]thiourea | MLS000587573 | SMR000211591 | [(Z)-[1-(4-fluorobenzyl)-2-keto-indolin-3-ylidene]amino]thiourea | [(Z)-[1-[(4-fluorophenyl)methyl]-2-oxo-3-indolylidene]amino]thiourea | [(Z)-[1-[(4-fluorophenyl)methyl]-2-oxoindol-3-ylidene]amino]thiourea | cid_6870780
TypeSmall organic molecule
Emp. Form.C16H13FN4OS
Mol. Mass.328.364
SMILESNC(=S)NN=C1C(=O)N(Cc2ccc(F)cc2)c2ccccc12 |w:4.3|
Structure
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