| Reaction Details |
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 | Report a problem with these data |
| Target | Ubiquitin-conjugating enzyme E2 N |
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| Ligand | BDBM79333 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay |
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| IC50 | 3607±161 nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Ubiquitin-conjugating enzyme E2 N |
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| Name: | Ubiquitin-conjugating enzyme E2 N |
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| Synonyms: | BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N |
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| Type: | PROTEIN |
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| Mol. Mass.: | 17137.61 |
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| Organism: | Homo sapiens (Human) |
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| Description: | EBI_101440 |
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| Residue: | 152 |
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| Sequence: | MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPE
EYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDP
LANDVAEQWKTNEAQAIETARAWTRLYAMNNI
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|
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| BDBM79333 |
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| n/a |
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| Name | BDBM79333 |
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| Synonyms: | MLS002391554 | SMR001355522 | [4-(8-hydroxy-6-quinolinyl)phenyl]-(1-piperazinyl)methanone;2,2,2-trifluoroacetic acid | [4-(8-hydroxy-6-quinolyl)phenyl]-piperazino-methanone;2,2,2-trifluoroacetic acid | [4-(8-hydroxyquinolin-6-yl)phenyl]-piperazin-1-ylmethanone;2,2,2-trifluoroacetic acid | [4-(8-oxidanylquinolin-6-yl)phenyl]-piperazin-1-yl-methanone;2,2,2-tris(fluoranyl)ethanoic acid | cid_44143204 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H19N3O2 |
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| Mol. Mass. | 333.3838 |
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| SMILES | Oc1cc(cc2cccnc12)-c1ccc(cc1)C(=O)N1CCNCC1 |
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| Structure | 
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