| Reaction Details |
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 | Report a problem with these data |
| Target | Perilipin-5 |
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| Ligand | BDBM34863 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain |
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| IC50 | 3408±n/a nM |
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| Citation |  PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) (2K validation set) PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Perilipin-5 |
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| Name: | Perilipin-5 |
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| Synonyms: | LSDP5 | OXPAT | PAT-1 | PLIN5 | PLIN5_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 50774.20 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_116292172 |
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| Residue: | 463 |
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| Sequence: | MSEEEAAQIPRSSVWEQDQQNVVQRVVALPLVRATCTAVCDVYSAAKDRHPLLGSACRLA
ENCVCGLTTRALDHAQPLLEHLQPQLATMNSLACRGLDKLEEKLPFLQQPSETVVTSAKD
VVASSVTGVVDLARRGRRWSVELKRSVSHAVDVVLEKSEELVDHFLPMTEEELAALAAEA
EGPEVGSVEDQRRQQGYFVRLGSLSARIRHLAYEHSVGKLRQSKHRAQDTLAQLQETLEL
IDHMQCGVTPTAPACPGKVHELWGEWGQRPPESRRRSQAELETLVLSRSLTQELQGTVEA
LESSVRGLPAGAQEKVAEVRRSVDALQTAFADARCFRDVPAAALAEGRGRVAHAHACVDE
LLELVVQAVPLPWLVGPFAPILVERPEPLPDLADLVDEVIGGPDPRWAHLDWPAQQRAWE
AEHRDGSGNGDGDRMGVAGDICEQEPETPSCPVKHTLMPELDF
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| BDBM34863 |
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| n/a |
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| Name | BDBM34863 |
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| Synonyms: | (5E)-5-(4,5-dimethoxy-2-nitro-benzylidene)-1-phenyl-barbituric acid | (5E)-5-[(4,5-dimethoxy-2-nitro-phenyl)methylidene]-1-phenyl-1,3-diazinane-2,4,6-trione | (5E)-5-[(4,5-dimethoxy-2-nitrophenyl)methylidene]-1-phenyl-1,3-diazinane-2,4,6-trione | 5-(4,5-dimethoxy-2-nitrobenzylidene)-1-phenyl-2,4,6(1H,3H,5H)-pyrimidinetrione | MLS000684314 | SMR000267903 | cid_1363391 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H15N3O7 |
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| Mol. Mass. | 397.3383 |
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| SMILES | COc1cc(C=C2C(=O)NC(=O)N(C2=O)c2ccccc2)c(cc1OC)[N+]([O-])=O |w:5.4| |
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| Structure | 
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