| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Perilipin-5 |
|---|
| Ligand | BDBM52777 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain |
|---|
| IC50 | 17555±n/a nM |
|---|
| Citation |  PubChem, PC Luminescence-based biochemical high throughput dose response assay for inhibitors of the interaction of the lipase co-activator protein, abhydrolase domain containing 5 (ABHD5) with perilipin-5 (MLDP; PLIN5) (2K validation set) PubChem Bioassay(2011)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Perilipin-5 |
|---|
| Name: | Perilipin-5 |
|---|
| Synonyms: | LSDP5 | OXPAT | PAT-1 | PLIN5 | PLIN5_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 50774.20 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_116292172 |
|---|
| Residue: | 463 |
|---|
| Sequence: | MSEEEAAQIPRSSVWEQDQQNVVQRVVALPLVRATCTAVCDVYSAAKDRHPLLGSACRLA
ENCVCGLTTRALDHAQPLLEHLQPQLATMNSLACRGLDKLEEKLPFLQQPSETVVTSAKD
VVASSVTGVVDLARRGRRWSVELKRSVSHAVDVVLEKSEELVDHFLPMTEEELAALAAEA
EGPEVGSVEDQRRQQGYFVRLGSLSARIRHLAYEHSVGKLRQSKHRAQDTLAQLQETLEL
IDHMQCGVTPTAPACPGKVHELWGEWGQRPPESRRRSQAELETLVLSRSLTQELQGTVEA
LESSVRGLPAGAQEKVAEVRRSVDALQTAFADARCFRDVPAAALAEGRGRVAHAHACVDE
LLELVVQAVPLPWLVGPFAPILVERPEPLPDLADLVDEVIGGPDPRWAHLDWPAQQRAWE
AEHRDGSGNGDGDRMGVAGDICEQEPETPSCPVKHTLMPELDF
|
|
|
|---|
| BDBM52777 |
|---|
| n/a |
|---|
| Name | BDBM52777 |
|---|
| Synonyms: | MLS000559965 | Methanesulfonic acid 3-oxo-2-[(E)-3-phenyl-prop-2-en-(Z)-ylidene]-2,3-dihydro-benzofuran-6-yl ester | SMR000439361 | [(2Z)-3-oxidanylidene-2-[(E)-3-phenylprop-2-enylidene]-1-benzofuran-6-yl] methanesulfonate | [(2Z)-3-oxo-2-[(E)-3-phenylprop-2-enylidene]-1-benzofuran-6-yl] methanesulfonate | cid_2015650 | methanesulfonic acid [(2Z)-3-keto-2-[(E)-3-phenylprop-2-enylidene]coumaran-6-yl] ester | methanesulfonic acid [(2Z)-3-oxo-2-[(E)-3-phenylprop-2-enylidene]-6-benzofuranyl] ester |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C18H14O5S |
|---|
| Mol. Mass. | 342.366 |
|---|
| SMILES | CS(=O)(=O)Oc1ccc2C(=O)\C(Oc2c1)=C\C=C\c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
