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TargetNorepinephrine transporter
LigandBDBM50014247
Substrate/Competitorn/a
Ki 121±n/a nM
CommentsPDSP_811
Citation Shank, RPVaught, JLPelley, KASetler, PEMcComsey, DFMaryanoff, BE McN-5652: a highly potent inhibitor of serotonin uptake. J Pharmacol Exp Ther247:1032-8 (1988) [PubMed]
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Norepinephrine transporter
Name:Norepinephrine transporter
Synonyms:n/a
Type:Enzyme Catalytic Domain
Mol. Mass.:2082.45
Organism:RAT
Description:Norepinephrine transporter 0 RAT::Q9JIA2
Residue:19
Sequence:
MLLARMKPQVQPELGGADQ
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BDBM50014247
n/a
NameBDBM50014247
Synonyms:(3R,4S)-3-(4-Methoxy-phenoxymethyl)-1-methyl-4-phenyl-piperidine | 3-(4-Methoxy-phenoxymethyl)-1-methyl-4-phenyl-piperidine(femoxetine) | CHEMBL94739 | Femoxetine
TypeSmall organic molecule
Emp. Form.C20H25NO2
Mol. Mass.311.418
SMILESCOc1ccc(OC[C@H]2CN(C)CC[C@@H]2c2ccccc2)cc1
Structure
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