| Reaction Details |
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 | Report a problem with these data |
| Target | Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
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| Ligand | BDBM49145 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay |
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| IC50 | 7473±540 nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS hits for Scp-1 phosphatase using a colorimetric assay PubChem Bioassay(2011)[AID] |
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| More Info.: | Get all data from this article, Assay Method |
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| Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
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| Name: | Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
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| Synonyms: | CTDS1_HUMAN | CTDSP1 | NIF3 | NLIIF | SCP1 | carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 isoform 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 29199.89 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_10864009 |
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| Residue: | 261 |
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| Sequence: | MDSSAVITQISKEEARGPLRGKGDQKSAASQKPRSRGILHSLFCCVCRDDGEALPAHSGA
PLLVEENGAIPKQTPVQYLLPEAKAQDSDKICVVIDLDETLVHSSFKPVNNADFIIPVEI
DGVVHQVYVLKRPHVDEFLQRMGELFECVLFTASLAKYADPVADLLDKWGAFRARLFRES
CVFHRGNYVKDLSRLGRDLRRVLILDNSPASYVFHPDNAVPVASWFDNMSDTELHDLLPF
FEQLSRVDDVYSVLRQPRPGS
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| BDBM49145 |
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| n/a |
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| Name | BDBM49145 |
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| Synonyms: | 6-(4-o-phenetylpiperazino)sulfonyl-1H-benzo[cd]indol-2-one | 6-[4-(2-ethoxyphenyl)piperazin-1-yl]sulfonyl-1H-benzo[cd]indol-2-one | 6-[[4-(2-ethoxyphenyl)-1-piperazinyl]sulfonyl]-1H-benzo[cd]indol-2-one | 6-{[4-(2-ethoxyphenyl)-1-piperazinyl]sulfonyl}benzo[cd]indol-2(1H)-one | MLS000049638 | SMR000076219 | cid_2133613 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H23N3O4S |
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| Mol. Mass. | 437.511 |
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| SMILES | CCOc1ccccc1N1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)c3cccc1c23 |
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| Structure | 
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