| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Thromboxane A2 receptor |
|---|
| Ligand | BDBM50010078 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_209599 |
|---|
| Kd | 6±n/a nM |
|---|
| Citation |  Misra, RN; Brown, BR; Han, WC; Harris, DN; Hedberg, A; Webb, ML; Hall, SE Interphenylene 7-oxabicyclo[2.2.1]heptane thromboxane A2 antagonists. Semicarbazone omega-chains. J Med Chem34:2882-91 (1991) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Thromboxane A2 receptor |
|---|
| Name: | Thromboxane A2 receptor |
|---|
| Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
|---|
| Type: | Enyzme |
|---|
| Mol. Mass.: | 37445.28 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P21731 |
|---|
| Residue: | 343 |
|---|
| Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
|
|
|
|---|
| BDBM50010078 |
|---|
| n/a |
|---|
| Name | BDBM50010078 |
|---|
| Synonyms: | CHEMBL95884 | [2-(5-oxabicyclo[2.2.1],3-formaldehyde (anilinocarbonyl)hydrazone-hept-2-ylmethyl)phenoxy]acetic acid |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H25N3O5 |
|---|
| Mol. Mass. | 423.4617 |
|---|
| SMILES | OC(=O)COc1ccccc1CC1C2CCC(O2)C1C=NNC(=O)Nc1ccccc1 |w:20.23,THB:11:12:17:15.14,19:18:17:15.14| |
|---|
| Structure | 
|
|---|
Search and Browse
