| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Adenosine receptor A1 |
|---|
| Ligand | BDBM50023502 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_28547 |
|---|
| IC50 | >10000±n/a nM |
|---|
| Citation |  Francis, JE; Cash, WD; Psychoyos, S; Ghai, G; Wenk, P; Friedmann, RC; Atkins, C; Warren, V; Furness, P; Hyun, JL Structure-activity profile of a series of novel triazoloquinazoline adenosine antagonists. J Med Chem31:1014-20 (1988) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Adenosine receptor A1 |
|---|
| Name: | Adenosine receptor A1 |
|---|
| Synonyms: | AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1 |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 36704.13 |
|---|
| Organism: | Rattus norvegicus (rat) |
|---|
| Description: | n/a |
|---|
| Residue: | 326 |
|---|
| Sequence: | MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGA
LVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVT
QRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYM
VYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALIL
FLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFL
KIWNDHFRCQPKPPIDEDLPEEKAED
|
|
|
|---|
| BDBM50023502 |
|---|
| n/a |
|---|
| Name | BDBM50023502 |
|---|
| Synonyms: | (9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)-dimethyl-amine | CHEMBL7759 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H12ClN5O |
|---|
| Mol. Mass. | 313.742 |
|---|
| SMILES | CN(C)c1nc2ccc(Cl)cc2c2nc(nn12)-c1ccco1 |
|---|
| Structure | 
|
|---|
Search and Browse
