Reaction Details |
| Report a problem with these data |
Target | Melatonin receptor type 1C |
---|
Ligand | BDBM50470702 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | ChEMBL_104611 (CHEMBL713590) |
---|
Ki | 350±n/a nM |
---|
Citation | Garratt, PJ; Jones, R; Tocher, DA; Sugden, D Mapping the melatonin receptor. 3. Design and synthesis of melatonin agonists and antagonists derived from 2-phenyltryptamines. J Med Chem38:1132-9 (1995) [PubMed] Article |
---|
More Info.: | Get all data from this article, Assay Method |
---|
|
Melatonin receptor type 1C |
---|
Name: | Melatonin receptor type 1C |
Synonyms: | CKB | MTR1C_CHICK | Mel-1C-R | Mel1c receptor | Melatonin receptor type 1C |
Type: | PROTEIN |
Mol. Mass.: | 38595.98 |
Organism: | Gallus gallus |
Description: | ChEMBL_104739 |
Residue: | 346 |
Sequence: | MERPGSNGSCSGCRLEGGPAARAASGLAAVLIVTIVVDVLGNALVILSVLRNKKLRNAGN
IFVVSLSVADLVVAVYPYPLILSAIFHNGWTMGNIHCQISGFLMGLSVIGSIFNITAIAI
NRYCYICHSLRYDKLFNLKNTCCYICLTWTLTVVAIVPNFFVGSLQYDPRIYSCTFAQTV
STSYTITVVVVHFIVPLSIVTFCYLRIWILVIQVKHRVRQDCKQKIRAADIRNFLTMFVV
FVLFAVCWGPLNFIGLAVSINPSKVQPHIPEWLFVLSYFMAYFNSCLNAVIYGLLNQNFR
KEYKRILLMLRTPRLLFIDVSKGGTEGLKSKPSPAVTNNNQAEIHL
|
|
|
BDBM50470702 |
---|
n/a |
---|
Name | BDBM50470702 |
Synonyms: | CHEMBL279188 |
Type | Small organic molecule |
Emp. Form. | C21H24N2O2 |
Mol. Mass. | 336.4275 |
SMILES | COCC(CNC(C)=O)c1c(-c2ccccc2)n(C)c2ccccc12 |
Structure |
|