| Reaction Details |
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 | Report a problem with these data |
| Target | Protein-glutamine gamma-glutamyltransferase, liver |
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| Ligand | BDBM81346 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_607926 (CHEMBL1066254) |
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| IC50 | 4000±n/a nM |
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| Citation |  Ozaki, S; Ebisui, E; Hamada, K; Goto, J; Suzuki, AZ; Terauchi, A; Mikoshiba, K Potent transglutaminase inhibitors, aryl beta-aminoethyl ketones. Bioorg Med Chem Lett20:1141-4 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Protein-glutamine gamma-glutamyltransferase, liver |
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| Name: | Protein-glutamine gamma-glutamyltransferase, liver |
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| Synonyms: | 2.3.2.13 | Protein-glutamine gamma-glutamyltransferase, liver |
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| Type: | PROTEIN |
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| Mol. Mass.: | 49544.80 |
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| Organism: | Cavia porcellus |
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| Description: | ChEMBL_109264 |
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| Residue: | 444 |
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| Sequence: | ILDICLMLLDTNPKFLKNAGQDCSRRSRPVYVGRVVSAMVNCNDDQGVLQGRWDNNYSDG
VSPMSWIGSVDILRRWKDYGCQRVKYGQCWVFAAVACTVLRCLAIPTRVVTNFNSAHDQN
SNLLIEYFRNESGEIEGNKSEMIWNFHSLLGGVVDDQAGPGAWVRGVQALDPTPQEKSEG
TYCCGPVPVRAIKEGHLNVKYDAPFVFAEVNADVVNWIRQKDGSLRKSINHLVVGLKIST
KSVGRDEREDITHTYKYPEGSEEEREAFVRANHLNKLATKEEAQEETGVAMRIRVGQNMT
MGSDFDIFAYITNGTAESHECQLLLCARIVSYNGVLGPVCSTNDLLNLTLDPFSENSIPL
HILYEKYGDYLTESNLIKVRGLLIEPAANSYVLAERDIYLENPEIKIRVLGEPKQNRKLI
AEVSLKNPLPVPLLGCIFTVEGAG
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| BDBM81346 |
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| n/a |
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| Name | BDBM81346 |
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| Synonyms: | CHEMBL538798 | M9440 (Me-3,4-dephostatin) |
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| Type | Small organic molecule |
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| Emp. Form. | C23H25NO |
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| Mol. Mass. | 331.4507 |
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| SMILES | CC(C)N(CCC(=O)c1ccc2ccccc2c1)Cc1ccccc1 |
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| Structure | 
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