| Reaction Details |
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 | Report a problem with these data |
| Target | Histamine H2 receptor |
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| Ligand | BDBM50483138 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_697529 (CHEMBL1638861) |
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| Ki | <1000±n/a nM |
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| Citation |  Igel, P; Dove, S; Buschauer, A Histamine H4 receptor agonists. Bioorg Med Chem Lett20:7191-9 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Histamine H2 receptor |
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| Name: | Histamine H2 receptor |
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| Synonyms: | Gastric receptor I | H2R | HISTAMINE H2 | HRH2 | HRH2_HUMAN | Histamine H2 receptor | Histamine H2-Gs alpha S |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 40115.31 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 359 |
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| Sequence: | MAPNGTASSFCLDSTACKITITVVLAVLILITVAGNVVVCLAVGLNRRLRNLTNCFIVSL
AITDLLLGLLVLPFSAIYQLSCKWSFGKVFCNIYTSLDVMLCTASILNLFMISLDRYCAV
MDPLRYPVLVTPVRVAISLVLIWVISITLSFLSIHLGWNSRNETSKGNHTTSKCKVQVNE
VYGLVDGLVTFYLPLLIMCITYYRIFKVARDQAKRINHISSWKAATIREHKATVTLAAVM
GAFIICWFPYFTAFVYRGLRGDDAINEVLEAIVLWLGYANSALNPILYAALNRDFRTGYQ
QLFCCRLANRNSHKTSLRSNASQLSRTQSREPRQQEEKPLKLQVWSGTEVTAPQGATDR
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| BDBM50483138 |
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| n/a |
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| Name | BDBM50483138 |
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| Synonyms: | CHEMBL1632414 |
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| Type | Small organic molecule |
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| Emp. Form. | C14H17ClN4O |
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| Mol. Mass. | 292.764 |
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| SMILES | CN1CCC(CC1)C(=N\O)\c1nc2cc(Cl)ccc2[nH]1 |
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| Structure | 
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