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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | D(2) dopamine receptor | ||
| Ligand | BDBM50055723 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | ChEMBL_62399 (CHEMBL872888) | ||
| Ki | 85±n/a nM | ||
| Citation |  Wustrow, DJ; Smith, WJ; Corbin, AE; Davis, MD; Georgic, LM; Pugsley, TA; Whetzel, SZ; Heffner, TG; Wise, LD 3-[[(4-Aryl-1-piperazinyl)alkyl]cyclohexyl]-1H-indoles as dopamine D2 partial agonists and autoreceptor agonists. J Med Chem40:250-9 (1997) [PubMed] Article | ||
| More Info.: | Get all data from this article, Assay Method | ||
| D(2) dopamine receptor | |||
| Name: | D(2) dopamine receptor | ||
| Synonyms: | DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2 | ||
| Type: | G Protein-Coupled Receptor (GPCR) | ||
| Mol. Mass.: | 50931.60 | ||
| Organism: | Rattus norvegicus (rat) | ||
| Description: | P61169 | ||
| Residue: | 444 | ||
| Sequence: |
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| BDBM50055723 | |||
| n/a | |||
| Name | BDBM50055723 | ||
| Synonyms: | 3-[4-(4-Pyridin-2-yl-piperazin-1-ylmethyl)-cyclohexyl]-1H-indole | CHEMBL87504 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C24H30N4 | ||
| Mol. Mass. | 374.5218 | ||
| SMILES | C([C@H]1CC[C@@H](CC1)c1c[nH]c2ccccc12)N1CCN(CC1)c1ccccn1 |wU:4.7,wD:1.0,(14,-4.05,;12.67,-4.82,;11.34,-4.05,;10.01,-4.82,;10.02,-6.35,;11.34,-7.12,;12.65,-6.36,;8.74,-7.2,;8.66,-8.74,;7.16,-9.15,;6.32,-7.87,;4.79,-7.64,;4.23,-6.19,;5.21,-4.98,;6.72,-5.23,;7.28,-6.65,;15.33,-4.82,;16.65,-4.02,;18,-4.79,;18.01,-6.33,;16.69,-7.12,;15.35,-6.36,;19.36,-7.09,;19.38,-8.63,;20.7,-9.38,;22.04,-8.6,;22.02,-7.06,;20.67,-6.3,)| | ||
| Structure | 
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