| Reaction Details |
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 | Report a problem with these data |
| Target | D(3) dopamine receptor |
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| Ligand | BDBM50523478 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1890410 (CHEMBL4392164) |
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| Ki | 3681±n/a nM |
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| Citation |  Keck, TM; Free, RB; Day, MM; Brown, SL; Maddaluna, MS; Fountain, G; Cooper, C; Fallon, B; Holmes, M; Stang, CT; Burkhardt, R; Bonifazi, A; Ellenberger, MP; Newman, AH; Sibley, DR; Wu, C; Boateng, CA Dopamine D J Med Chem62:3722-3740 (2019) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(3) dopamine receptor |
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| Name: | D(3) dopamine receptor |
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| Synonyms: | DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3 |
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| Type: | n/a |
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| Mol. Mass.: | 44243.43 |
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| Organism: | Homo sapiens (Human) |
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| Description: | n/a |
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| Residue: | 400 |
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| Sequence: | MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERAL
QTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILN
LCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTV
CSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQ
QTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRK
LSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHV
SPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
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| BDBM50523478 |
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| n/a |
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| Name | BDBM50523478 |
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| Synonyms: | CHEMBL4473792 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H26N2O |
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| Mol. Mass. | 322.4439 |
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| SMILES | Cc1ccc(cc1)C1CCN(CC(=O)Nc2cccc(C)c2)CC1 |
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| Structure | 
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