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TargetCoagulation factor VII
LigandBDBM50127212
Substrate/Competitorn/a
Meas. Tech.ChEMBL_48461 (CHEMBL663024)
IC50 2±n/a nM
Citation Zobel, KKoehler, MFBeresini, MHCaris, LDCombs, D Phosphate ester serum albumin affinity tags greatly improve peptide half-life in vivo. Bioorg Med Chem Lett13:1513-5 (2003) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Coagulation factor VII
Name:Coagulation factor VII
Synonyms:Eptacog alfa | F7 | FA7_HUMAN | Factor VIIa | Factor VIIa (fVIIa) | Proconvertin | SPCA | Thrombin and coagulation factor VII | serum prothrombin conversion accelerator
Type:Enzyme
Mol. Mass.:51599.89
Organism:Homo sapiens (Human)
Description:n/a
Residue:466
Sequence:
MVSQALRLLCLLLGLQGCLAAGGVAKASGGETRDMPWKPGPHRVFVTQEEAHGVLHRRRR
ANAFLEELRPGSLERECKEEQCSFEEAREIFKDAERTKLFWISYSDGDQCASSPCQNGGS
CKDQLQSYICFCLPAFEGRNCETHKDDQLICVNENGGCEQYCSDHTGTKRSCRCHEGYSL
LADGVSCTPTVEYPCGKIPILEKRNASKPQGRIVGGKVCPKGECPWQVLLLVNGAQLCGG
TLINTIWVVSAAHCFDKIKNWRNLIAVLGEHDLSEHDGDEQSRRVAQVIIPSTYVPGTTN
HDIALLRLHQPVVLTDHVVPLCLPERTFSERTLAFVRFSLVSGWGQLLDRGATALELMVL
NVPRLMTQDCLQQSRKVGDSPNITEYMFCAGYSDGSKDSCKGDSGGPHATHYRGTWYLTG
IVSWGQGCATVGHFGVYTRVSQYIEWLQKLMRSEPRPGVLLRAPFP
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50127212
n/a
NameBDBM50127212
Synonyms:ALCDNPRIDRWYCQFVEG peptide analogue | CHEMBL2372335
TypeSmall organic molecule
Emp. Form.C112H157N28O32PS2
Mol. Mass.2502.717
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Structure
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