| Reaction Details |
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 | Report a problem with these data |
| Target | Serine protease 1 |
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| Ligand | BDBM50141562 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_213081 |
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| Ki | 32000±n/a nM |
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| Citation |  Zega, A; Mlinsek, G; Solmajer, T; Trampus-Bakija, A; Stegnar, M; Urleb, U Thrombin inhibitors built on an azaphenylalanine scaffold. Bioorg Med Chem Lett14:1563-7 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Serine protease 1 |
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| Name: | Serine protease 1 |
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| Synonyms: | Alpha-trypsin chain 1 | Alpha-trypsin chain 2 | Beta-trypsin | Cationic trypsinogen | PRSS1 | Serine protease 1 | TRP1 | TRY1 | TRY1_HUMAN | TRYP1 | Thrombin & trypsin | Trypsin | Trypsin I | Trypsin-1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 26557.80 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P07477 |
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| Residue: | 247 |
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| Sequence: | MNPLLILTFVAAALAAPFDDDDKIVGGYNCEENSVPYQVSLNSGYHFCGGSLINEQWVVS
AGHCYKSRIQVRLGEHNIEVLEGNEQFINAAKIIRHPQYDRKTLNNDIMLIKLSSRAVIN
ARVSTISLPTAPPATGTKCLISGWGNTASSGADYPDELQCLDAPVLSQAKCEASYPGKIT
SNMFCVGFLEGGKDSCQGDSGGPVVCNGQLQGVVSWGDGCAQKNKPGVYTKVYNYVKWIK
NTIAANS
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| BDBM50141562 |
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| n/a |
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| Name | BDBM50141562 |
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| Synonyms: | Azaphenylalanine derivative | CHEMBL39078 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H29N5O4S |
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| Mol. Mass. | 495.594 |
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| SMILES | ONC(=N)c1cccc(CN(NS(=O)(=O)c2ccc3ccccc3c2)C(=O)N2CCCCCC2)c1 |
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| Structure | 
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