| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50150797 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_305297 (CHEMBL832845) |
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| IC50 | >10000±n/a nM |
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| Citation |  Balboni, G; Salvadori, S; Guerrini, R; Negri, L; Giannini, E; Bryant, SD; Jinsmaa, Y; Lazarus, LH Direct influence of C-terminally substituted amino acids in the Dmt-Tic pharmacophore on delta-opioid receptor selectivity and antagonism. J Med Chem47:4066-71 (2004) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
|
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|
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| BDBM50150797 |
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| n/a |
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| Name | BDBM50150797 |
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| Synonyms: | 2-[2-Amino-3-((S)-4-hydroxy-2,6-dimethyl-phenyl)-propionyl]-1,2,3,4-tetrahydro-isoquinoline-3-carboxylic acid (1-carbamoyl-ethyl)-amide | CHEMBL359786 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H30N4O4 |
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| Mol. Mass. | 438.5194 |
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| SMILES | C[C@H](NC(=O)C1Cc2ccccc2CN1C(=O)C(N)Cc1c(C)cc(O)cc1C)C(N)=O |
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| Structure | 
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