| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Pyroglutamylated RF-amide peptide receptor |
|---|
| Ligand | BDBM50583773 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_2158121 (CHEMBL5042871) |
|---|
| Ki | >50000±n/a nM |
|---|
| Citation |  Quillet, R; Schneider, S; Utard, V; Drieu la Rochelle, A; Elhabazi, K; Henningsen, JB; Gizzi, P; Schmitt, M; Kugler, V; Simonneaux, V; Ilien, B; Simonin, F; Bihel, F Identification of an J Med Chem64:7555-7564 (2021) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Pyroglutamylated RF-amide peptide receptor |
|---|
| Name: | Pyroglutamylated RF-amide peptide receptor |
|---|
| Synonyms: | GPR103 | Pyroglutamylated RFamide peptide receptor | QRFPR | QRFPR_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 49508.46 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | GPR103 0 HUMAN::Q96P65 |
|---|
| Residue: | 431 |
|---|
| Sequence: | MQALNITPEQFSRLLRDHNLTREQFIALYRLRPLVYTPELPGRAKLALVLTGVLIFALAL
FGNALVFYVVTRSKAMRTVTNIFICSLALSDLLITFFCIPVTMLQNISDNWLGGAFICKM
VPFVQSTAVVTEILTMTCIAVERHQGLVHPFKMKWQYTNRRAFTMLGVVWLVAVIVGSPM
WHVQQLEIKYDFLYEKEHICCLEEWTSPVHQKIYTTFILVILFLLPLMVMLILYSKIGYE
LWIKKRVGDGSVLRTIHGKEMSKIARKKKRAVIMMVTVVALFAVCWAPFHVVHMMIEYSN
FEKEYDDVTIKMIFAIVQIIGFSNSICNPIVYAFMNENFKKNVLSAVCYCIVNKTFSPAQ
RHGNSGITMMRKKAKFSLRENPVEETKGEAFSDGNIEVKLCEQTEEKKKLKRHLALFRSE
LAENSPLDSGH
|
|
|
|---|
| BDBM50583773 |
|---|
| n/a |
|---|
| Name | BDBM50583773 |
|---|
| Synonyms: | CHEMBL5091013 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C23H28N6O3 |
|---|
| Mol. Mass. | 436.5068 |
|---|
| SMILES | [#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]-[#7]-[#6](-[#7])=[#7])-[#7]-[#6](=O)\[#6]=[#6](\c1ccccc1)-c1ccccc1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
