| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Glucose-dependent insulinotropic receptor |
|---|
| Ligand | BDBM50610721 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_2281774 |
|---|
| IC50 | 18400±n/a nM |
|---|
| Citation |  Alizadeh, SR; Ebrahimzadeh, MA Pyrazolotriazines: Biological activities, synthetic strategies and recent developments. Eur J Med Chem223:0 (2021) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Glucose-dependent insulinotropic receptor |
|---|
| Name: | Glucose-dependent insulinotropic receptor |
|---|
| Synonyms: | G-protein coupled receptor 119 (GPR119) | GP119_HUMAN | GPR119 | Glucose-dependent insulinotropic receptor |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 36901.49 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q8TDV5 |
|---|
| Residue: | 335 |
|---|
| Sequence: | MESSFSFGVILAVLASLIIATNTLVAVAVLLLIHKNDGVSLCFTLNLAVADTLIGVAISG
LLTDQLSSPSRPTQKTLCSLRMAFVTSSAAASVLTVMLITFDRYLAIKQPFRYLKIMSGF
VAGACIAGLWLVSYLIGFLPLGIPMFQQTAYKGQCSFFAVFHPHFVLTLSCVGFFPAMLL
FVFFYCDMLKIASMHSQQIRKMEHAGAMAGGYRSPRTPSDFKALRTVSVLIGSFALSWTP
FLITGIVQVACQECHLYLVLERYLWLLGVGNSLLNPLIYAYWQKEVRLQLYHMALGVKKV
LTSFLLFLSARNCGPERPRESSCHIVTISSSEFDG
|
|
|
|---|
| BDBM50610721 |
|---|
| n/a |
|---|
| Name | BDBM50610721 |
|---|
| Synonyms: | CHEMBL5271736 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H13FN6 |
|---|
| Mol. Mass. | 320.3237 |
|---|
| SMILES | Nc1nc(Nc2ccc(F)cc2)n2nc(cc2n1)-c1ccccc1 |
|---|
| Structure | 
|
|---|
Search and Browse
