| Reaction Details |
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 | Report a problem with these data |
| Target | Phospholipase A2 |
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| Ligand | BDBM50263053 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_489269 (CHEMBL990825) |
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| IC50 | >320±n/a nM |
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| Citation |  Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem51:4708-14 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Phospholipase A2 |
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| Name: | Phospholipase A2 |
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| Synonyms: | PA21B_MOUSE | Phospholipase A2 group 1B | Pla2 | Pla2g1b |
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| Type: | PROTEIN |
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| Mol. Mass.: | 16291.94 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_489269 |
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| Residue: | 146 |
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| Sequence: | MKLLLLAALLTAGAAAHSISPRAVWQFRNMIKCTIPGSDPLKDYNNYGCYCGLGGWGTPV
DDLDRCCQTHDHCYSQAKKLESCKFLIDNPYTNTYSYSCSGSEITCSAKNNKCEDFICNC
DREAAICFSKVPYNKEYKNLDTGKFC
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| BDBM50263053 |
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| n/a |
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| Name | BDBM50263053 |
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| Synonyms: | 2-(3-Biphenyl-2-ylmethyl-2-ethyl-8-methoxy-indolizin-1-yl)-2-oxo-acetamide | CHEMBL478821 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H24N2O3 |
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| Mol. Mass. | 412.4804 |
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| SMILES | CCc1c(Cc2ccccc2-c2ccccc2)n2cccc(OC)c2c1C(=O)C(N)=O |
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| Structure | 
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