Reaction Details |
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Target | Thromboxane A2 receptor |
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Ligand | BDBM50047266 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEBML_209598 |
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Kd | 0.100000±n/a nM |
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Citation | Misra, RN; Harris, DN; Michel, IM; Goldenberg, HJ; Webb, ML; Brown, BR Interphenylene phenyl oxazoles: novel, potent thromboxane receptor antagonists Bioorg Med Chem Lett2:937-940 (1992) Article |
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More Info.: | Get all data from this article, Assay Method |
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Thromboxane A2 receptor |
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Name: | Thromboxane A2 receptor |
Synonyms: | Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta |
Type: | Enyzme |
Mol. Mass.: | 37445.28 |
Organism: | Homo sapiens (Human) |
Description: | P21731 |
Residue: | 343 |
Sequence: | MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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BDBM50047266 |
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n/a |
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Name | BDBM50047266 |
Synonyms: | 3-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-yl]-7-oxa-bicyclo[2.2.1]hept-2-ylmethyl}-phenyl)-propionic acid | CHEMBL31765 |
Type | Small organic molecule |
Emp. Form. | C30H40N2O5 |
Mol. Mass. | 508.649 |
SMILES | OC(=O)CCc1ccccc1CC1C2CCC(O2)C1c1nc(co1)C(=O)NCCCCC1CCCCC1 |THB:19:18:17:15.14,11:12:17:15.14| |
Structure |
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