| Reaction Details |
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 | Report a problem with these data |
| Target | Cholecystokinin receptor type A |
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| Ligand | BDBM50281728 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_50203 |
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| IC50 | 20000±n/a nM |
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| Citation |  Bock, MG; DiPardo, RM; Veber, DF; Chang, RS; Lotti, VJ; Freedman, SB; Freidinger, RM Benzolactams as non-peptide cholecystokinin receptor ligands Bioorg Med Chem Lett3:871-874 (1993) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cholecystokinin receptor type A |
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| Name: | Cholecystokinin receptor type A |
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| Synonyms: | CCKAR_RAT | Cckar | Cholecystokinin peripheral | Cholecystokinin receptor | Cholecystokinin receptor type A |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 49676.37 |
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| Organism: | RAT |
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| Description: | Cholecystokinin central 0 RAT::P30551 |
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| Residue: | 444 |
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| Sequence: | MSHSPARQHLVESSRMDVVDSLLMNGSNITPPCELGLENETLFCLDQPQPSKEWQSALQI
LLYSIIFLLSVLGNTLVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPNLLK
DFIFGSAVCKTTTYFMGTSVSVSTFNLVAISLERYGAICRPLQSRVWQTKSHALKVIAAT
WCLSFTIMTPYPIYSNLVPFTKNNNQTANMCRFLLPSDAMQQSWQTFLLLILFLLPGIVM
VVAYGLISLELYQGIKFDASQKKSAKEKKPSTGSSTRYEDSDGCYLQKSRPPRKLELQQL
SSGSGGSRLNRIRSSSSAANLIAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAE
KHLSGTPISFILLLSYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGPPGVRGEVGEEE
DGRTIRALLSRYSYSHMSTSAPPP
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| BDBM50281728 |
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| n/a |
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| Name | BDBM50281728 |
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| Synonyms: | CHEMBL170068 | [3-(3-Naphthalen-1-yl-ureido)-2-oxo-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl]-acetic acid |
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| Type | Small organic molecule |
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| Emp. Form. | C23H21N3O4 |
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| Mol. Mass. | 403.4305 |
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| SMILES | OC(=O)CN1c2ccccc2CCC(NC(=O)Nc2cccc3ccccc23)C1=O |
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| Structure | 
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