| Reaction Details |
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 | Report a problem with these data |
| Target | Cytosol aminopeptidase |
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| Ligand | BDBM50022754 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_98398 |
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| Ki | 26000±n/a nM |
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| Citation |  Ocain, TD; Rich, DH Synthesis of sulfur-containing analogues of bestatin. Inhibition of aminopeptidases by alpha-thiolbestatin analogues. J Med Chem31:2193-9 (1988) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Cytosol aminopeptidase |
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| Name: | Cytosol aminopeptidase |
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| Synonyms: | AMPL_HUMAN | Aminopeptidase | LAP3 | LAPEP | Leucine aminopeptidase | PEPS |
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| Type: | PROTEIN |
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| Mol. Mass.: | 56171.75 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1507539 |
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| Residue: | 519 |
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| Sequence: | MFLLPLPAAGRVVVRRLAVRRFGSRSLSTADMTKGLVLGIYSKEKEDDVPQFTSAGENFD
KLLAGKLRETLNISGPPLKAGKTRTFYGLHQDFPSVVLVGLGKKAAGIDEQENWHEGKEN
IRAAVAAGCRQIQDLELSSVEVDPCGDAQAAAEGAVLGLYEYDDLKQKKKMAVSAKLYGS
GDQEAWQKGVLFASGQNLARQLMETPANEMTPTRFAEIIEKNLKSASSKTEVHIRPKSWI
EEQAMGSFLSVAKGSDEPPVFLEIHYKGSPNANEPPLVFVGKGITFDSGGISIKASANMD
LMRADMGGAATICSAIVSAAKLNLPINIIGLAPLCENMPSGKANKPGDVVRAKNGKTIQV
DNTDAEGRLILADALCYAHTFNPKVILNAATLTGAMDVALGSGATGVFTNSSWLWNKLFE
ASIETGDRVWRMPLFEHYTRQVVDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHL
DIAGVMTNKDEVPYLRKGMTGRPTRTLIEFLLRFSQDNA
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| BDBM50022754 |
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| n/a |
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| Name | BDBM50022754 |
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| Synonyms: | 3-Amino-2-mercapto-N-(3-methyl-butyl)-4-phenyl-butyramide | CHEMBL69238 |
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| Type | Small organic molecule |
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| Emp. Form. | C15H24N2OS |
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| Mol. Mass. | 280.429 |
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| SMILES | CC(C)CCNC(=O)[C@H](S)[C@@H](N)Cc1ccccc1 |
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| Structure | 
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