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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50359499
Substrate/Competitorn/a
Meas. Tech.ChEBML_201270
Ki 8320±n/a nM
Citation Glennon, RASmith, JDIsmaiel, AMel-Ashmawy, MBattaglia, GFischer, JB Identification and exploitation of the sigma-opiate pharmacophore. J Med Chem34:1094-8 (1991) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Aging-associated gene 8 protein | OPRS1 | SGMR1_HUMAN | SIG-1R | SIGMAR1 | SR-BP | SR31747-binding protein | SRBP | Sigma 1-type opioid receptor | Sigma opioid receptor | Sigma1R | hSigmaR1
Type:Enzyme Catalytic Domain
Mol. Mass.:25124.85
Organism:Homo sapiens (Human)
Description:Q99720
Residue:223
Sequence:
MQWAVGRRWAWAALLLAVAAVLTQVVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSRGHSGRY
WAEISDTIISGTFHQWREGTTKSEVFYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALADTVFSTQDFLTLFYTLRSYARGLRLELTTYLFGQDP
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BDBM50359499
n/a
NameBDBM50359499
Synonyms:(S)Methamphetamine | METHAMPHETAMINE
TypeSmall organic molecule
Emp. Form.C10H15N
Mol. Mass.149.2328
SMILESCN[C@@H](C)Cc1ccccc1 |r|
Structure
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