| Reaction Details |
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 | Report a problem with these data |
| Target | Adenosine receptor A2a |
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| Ligand | BDBM50453916 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_30929 (CHEMBL647738) |
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| Ki | 22100±n/a nM |
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| Citation |  van der Wenden, EM; von Frijtag Drabbe Künzel, JK; Mathôt, RA; Danhof, M; IJzerman, AP; Soudijn, W Ribose-modified adenosine analogues as potential partial agonists for the adenosine receptor. J Med Chem38:4000-6 (1995) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Adenosine receptor A2a |
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| Name: | Adenosine receptor A2a |
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| Synonyms: | AA2AR_RAT | ADENOSINE A2a | Adenosine A2 receptor | Adenosine A2a receptor (A2a) | Adenosine Receptors A2a (A2a) | Adenosine receptor A2a and A3 | Adenosine receptors A2a | Adora2a | Rat striatal adenosine A2a receptor |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 45015.65 |
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| Organism: | Rattus norvegicus (rat) |
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| Description: | Rat A2A receptors expressed in CHO cells. |
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| Residue: | 410 |
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| Sequence: | MGSSVYITVELAIAVLAILGNVLVCWAVWINSNLQNVTNFFVVSLAAADIAVGVLAIPFA
ITISTGFCAACHGCLFFACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGVRAKG
IIAICWVLSFAIGLTPMLGWNNCSQKDGNSTKTCGEGRVTCLFEDVVPMNYMVYYNFFAF
VLLPLLLMLAIYLRIFLAARRQLKQMESQPLPGERTRSTLQKEVHAAKSLAIIVGLFALC
WLPLHIINCFTFFCSTCRHAPPWLMYLAIILSHSNSVVNPFIYAYRIREFRQTFRKIIRT
HVLRRQEPFQAGGSSAWALAAHSTEGEQVSLRLNGHPLGVWANGSATHSGRRPNGYTLGL
GGGGSAQGSPRDVELPTQERQEGQEHPGLRGHLVQARVGASSWSSEFAPS
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| BDBM50453916 |
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| n/a |
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| Name | BDBM50453916 |
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| Synonyms: | CHEMBL2112665 |
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| Type | Small organic molecule |
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| Emp. Form. | C16H23N5O3 |
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| Mol. Mass. | 333.3855 |
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| SMILES | OC[C@@H]1C[C@@H](O)[C@@H](O1)n1cnc2c(NC3CCCCC3)ncnc12 |r| |
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| Structure | 
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