Reaction Details |
![](/images/Email.png) | Report a problem with these data |
Target | Somatostatin receptor type 5 |
---|
Ligand | BDBM50423465 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | ChEMBL_461991 (CHEMBL944834) |
---|
Kd | 56234±n/a nM |
---|
Citation | Troxler, T; Enz, A; Hoyer, D; Langenegger, D; Neumann, P; Pfäffli, P; Schoeffter, P; Hurth, K Ergoline derivatives as highly potent and selective antagonists at the somatostatin sst 1 receptor. Bioorg Med Chem Lett18:979-82 (2008) [PubMed] Article |
---|
More Info.: | Get all data from this article, Assay Method |
---|
|
Somatostatin receptor type 5 |
---|
Name: | Somatostatin receptor type 5 |
Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
Type: | Enzyme |
Mol. Mass.: | 39218.02 |
Organism: | Homo sapiens (Human) |
Description: | P35346 |
Residue: | 364 |
Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
|
|
|
BDBM50423465 |
---|
n/a |
---|
Name | BDBM50423465 |
Synonyms: | ERGOLINE |
Type | Small organic molecule |
Emp. Form. | C26H30BrN5O2 |
Mol. Mass. | 524.453 |
SMILES | CN1C[C@@H](C[C@H]2[C@H]1Cc1c(Br)[nH]c3cccc2c13)C(=O)N1CCN(CC1)c1cccc(=O)n1C |
Structure |
|