| Reaction Details |
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 | Report a problem with these data |
| Target | Free fatty acid receptor 1 |
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| Ligand | BDBM50434295 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1585169 (CHEMBL3820977) |
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| EC50 | 19±n/a nM |
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| Citation |  Christiansen, E; Hudson, BD; Hansen, AH; Milligan, G; Ulven, T Development and Characterization of a Potent Free Fatty Acid Receptor 1 (FFA1) Fluorescent Tracer. J Med Chem59:4849-58 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Free fatty acid receptor 1 |
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| Name: | Free fatty acid receptor 1 |
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| Synonyms: | FFAR1 | FFAR1_HUMAN | G-protein Coupled Receptor 40 | GPR40 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 31473.32 |
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| Organism: | Homo sapiens (Human) |
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| Description: | O14842 |
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| Residue: | 300 |
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| Sequence: | MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSLVYALNLGCSDLLLTVSLP
LKAVEALASGAWPLPASLCPVFAVAHFFPLYAGGGFLAALSAGRYLGAAFPLGYQAFRRP
CYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAG
PARFSLSLLLFFLPLAITAFCYVGCLRALARSGLTHRRKLRAAWVAGGALLTLLLCVGPY
NASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLGRGPGLKTVCAARTQGGKSQK
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| BDBM50434295 |
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| n/a |
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| Name | BDBM50434295 |
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| Synonyms: | CHEMBL2386353 |
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| Type | Small organic molecule |
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| Emp. Form. | C19H14FNO2 |
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| Mol. Mass. | 307.3184 |
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| SMILES | OC(=O)CCc1ccc(cc1F)C#Cc1ccccc1CC#N |
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| Structure | 
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