| Reaction Details |
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 | Report a problem with these data |
| Target | D(4) dopamine receptor |
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| Ligand | BDBM50182751 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1586515 (CHEMBL3821454) |
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| Ki | 123±n/a nM |
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| Citation |  Ofori, E; Zhu, XY; Etukala, JR; Peprah, K; Jordan, KR; Adkins, AA; Bricker, BA; Kang, HJ; Huang, XP; Roth, BL; Ablordeppey, SY Design and synthesis of dual 5-HT1A and 5-HT7 receptor ligands. Bioorg Med Chem24:3464-71 (2016) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| D(4) dopamine receptor |
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| Name: | D(4) dopamine receptor |
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| Synonyms: | D(4) dopamine receptor | DOPAMINE D4 | DOPAMINE D4.4 | DRD4_RAT | Dopamine receptor | Drd4 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41307.65 |
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| Organism: | RAT |
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| Description: | DOPAMINE D4.4 0 RAT::P30729 |
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| Residue: | 387 |
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| Sequence: | MGNSSATGDGGLLAGRGPESLGTGTGLGGAGAAALVGGVLLIGMVLAGNSLVCVSVASER
ILQTPTNYFIVSLAAADLLLAVLVLPLFVYSEVQGGVWLLSPRLCDTLMAMDVMLCTASI
FNLCAISVDRFVAVTVPLRYNQQGQCQLLLIAATWLLSAAVAAPVVCGLNDVPGRDPTVC
CLEDRDYVVYSSICSFFLPCPLMLLLYWATFRGLRRWEAARHTKLHSRAPRRPSGPGPPV
SDPTQGPLFSDCPPPSPSLRTSPTVSSRPESDLSQSPCSPGCLLPDAALAQPPAPSSRRK
RGAKITGRERKAMRVLPVVVGAFLMCWTPFFVVHITRALCPACFVSPRLVSAVTWLGYVN
SALNPIIYTIFNAEFRSVFRKTLRLRC
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| BDBM50182751 |
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| n/a |
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| Name | BDBM50182751 |
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| Synonyms: | CHEMBL3819082 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H23ClFN |
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| Mol. Mass. | 331.855 |
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| SMILES | Cl.Fc1ccc2CC(CCN3CCc4ccccc4C3)Cc2c1 |
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| Structure | 
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