Reaction Details |
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Target | Delta-type opioid receptor |
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Ligand | BDBM50128080 |
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Substrate/Competitor | n/a |
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Ki | 1.5±n/a nM |
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Comments | PDSP_772 |
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Citation | Toll, L; Berzetei-Gurske, IP; Polgar, WE; Brandt, SR; Adapa, ID; Rodriguez, L; Schwartz, RW; Haggart, D; O'Brien, A; White, A; Kennedy, JM; Craymer, K; Farrington, L; Auh, JS Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA Res Monogr178:440-66 (1998) [PubMed] |
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More Info.: | Get all data from this article |
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Delta-type opioid receptor |
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Name: | Delta-type opioid receptor |
Synonyms: | Delta opioid receptor | Delta-type opioid receptor | OPIATE Delta | OPRD1 | OPRD_PIG |
Type: | Enzyme Catalytic Domain |
Mol. Mass.: | 25736.90 |
Organism: | GUINEA PIG |
Description: | OPIATE Delta OPRD1 GUINEA PIG::P79291 |
Residue: | 228 |
Sequence: | GIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNM
FTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPR
DGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILVITVCYGLMLLRLRSVRLLSGSKEK
DRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAAL
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BDBM50128080 |
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n/a |
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Name | BDBM50128080 |
Synonyms: | CHEMBL217379 | DYNORPHIN(1-8)-OH | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-OH |
Type | Small organic molecule |
Emp. Form. | C46H72N14O10 |
Mol. Mass. | 981.1517 |
SMILES | CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(O)=O |
Structure |
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