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TargetCorticotropin-releasing factor-binding protein
LigandBDBM46468
Substrate/Competitorn/a
Meas. Tech.Dose Response confirmation of uHTS hits for small molecule agonists of the CRF-binding protein and CRF-R2 receptor complex
EC50>53000±n/a nM
Citation PubChem, PC Dose Response confirmation of uHTS hits for small molecule agonists of the CRF-binding protein and CRF-R2 receptor complex PubChem Bioassay(2012)[AID]
More Info.:Get all data from this article,  Assay Method
 
Corticotropin-releasing factor-binding protein
Name:Corticotropin-releasing factor-binding protein
Synonyms:CRFBP | CRHBP | CRHBP_HUMAN | corticotropin releasing factor-binding protein
Type:Enzyme Catalytic Domain
Mol. Mass.:36143.95
Organism:Homo sapiens (Human)
Description:P24387
Residue:322
Sequence:
MSPNFKLQCHFILIFLTALRGESRYLELREAADYDPFLLFSANLKRELAGEQPYRRALRC
LDMLSLQGQFTFTADRPQLHCAAFFISEPEEFITIHYDQVSIDCQGGDFLKVFDGWILKG
EKFPSSQDHPLPSAERYIDFCESGLSRRSIRSSQNVAMIFFRVHEPGNGFTLTIKTDPNL
FPCNVISQTPNGKFTLVVPHQHRNCSFSIIYPVVIKISDLTLGHVNGLQLKKSSAGCEGI
GDFVELLGGTGLDPSKMTPLADLCYPFHGPAQMKVGCDNTVVRMVSSGKHVNRVTFEYRQ
LEPYELENPNGNSIGEFCLSGL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM46468
n/a
NameBDBM46468
Synonyms:3-[allyl(phenyl)sulfamoyl]benzoic acid | 3-[phenyl(prop-2-enyl)sulfamoyl]benzoic acid | MLS000570026 | SMR000150082 | cid_2386003
TypeSmall organic molecule
Emp. Form.C16H15NO4S
Mol. Mass.317.36
SMILESOC(=O)c1cccc(c1)S(=O)(=O)N(CC=C)c1ccccc1
Structure
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