| Reaction Details |
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 | Report a problem with these data |
| Target | Corticotropin-releasing factor-binding protein |
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| Ligand | BDBM90193 |
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| Substrate/Competitor | n/a |
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| IC50 | 4960±n/a nM |
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| Citation |  PubChem, PC Dose Response confirmation of uHTS hits for small molecule antagonists of the CRF-binding protein and CRF-R2 receptor complex in 384 well format PubChem Bioassay(2012)[AID] |
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| More Info.: | Get all data from this article |
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| Corticotropin-releasing factor-binding protein |
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| Name: | Corticotropin-releasing factor-binding protein |
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| Synonyms: | CRFBP | CRHBP | CRHBP_HUMAN | corticotropin releasing factor-binding protein |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 36143.95 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P24387 |
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| Residue: | 322 |
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| Sequence: | MSPNFKLQCHFILIFLTALRGESRYLELREAADYDPFLLFSANLKRELAGEQPYRRALRC
LDMLSLQGQFTFTADRPQLHCAAFFISEPEEFITIHYDQVSIDCQGGDFLKVFDGWILKG
EKFPSSQDHPLPSAERYIDFCESGLSRRSIRSSQNVAMIFFRVHEPGNGFTLTIKTDPNL
FPCNVISQTPNGKFTLVVPHQHRNCSFSIIYPVVIKISDLTLGHVNGLQLKKSSAGCEGI
GDFVELLGGTGLDPSKMTPLADLCYPFHGPAQMKVGCDNTVVRMVSSGKHVNRVTFEYRQ
LEPYELENPNGNSIGEFCLSGL
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| BDBM90193 |
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| n/a |
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| Name | BDBM90193 |
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| Synonyms: | MLS000335120 | N-[1-(1H-benzimidazol-2-yl)-2-phenyl-ethyl]-4-chloranyl-3-nitro-benzamide | N-[1-(1H-benzimidazol-2-yl)-2-phenyl-ethyl]-4-chloro-3-nitro-benzamide | N-[1-(1H-benzimidazol-2-yl)-2-phenylethyl]-4-chloro-3-nitrobenzamide | SMR000249878 | cid_3320062 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H17ClN4O3 |
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| Mol. Mass. | 420.848 |
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| SMILES | [O-][N+](=O)c1cc(ccc1Cl)C(=O)NC(Cc1ccccc1)c1nc2ccccc2[nH]1 |
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| Structure | 
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