| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 2A |
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| Ligand | BDBM114603 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Late stage for the probe development effort to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) |
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| EC50 | 76083±n/a nM |
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| Citation |  PubChem, PC Late stage for the probe development effort to identify agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A): Luminescence-based cell-based high throughput dose response assay for agonists of the mouse 5-hydroxytryptamine (serotonin) receptor 2A (HTR2A) PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| 5-hydroxytryptamine receptor 2A |
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| Name: | 5-hydroxytryptamine receptor 2A |
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| Synonyms: | 5-HT-2 | 5-HT-2A | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A (5HT2A) | 5HT2A_MOUSE | Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor | Htr2 | Htr2a | Serotonin 2a (5-HT2a) receptor |
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| Type: | Enzyme |
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| Mol. Mass.: | 52843.00 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | P35363 |
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| Residue: | 471 |
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| Sequence: | MEILCEDNISLSSIPNSLMQLGDDSRLYPNDFNSRDANTSEASNWTIDAENRTNLSCEGY
LPPTCLSILHLQEKNWSALLTTVVIILTIAGNILVIMAVSLEKKLQNATNYFLMSLAIAD
MLLGFLVMPVSMLTILYGYRWPLPSKLCAVWIYLDVLFSTASIMHLCAISLDRYVAIQNP
IHHSRFNSRTKAFLKIIAVWTISVGISMPIPVFGLQDDSKVFKEGSCLLADDNFVLIGSF
VAFFIPLTIMVITYFLTIKSLQKEATLCVSDLSTRAKLSSFSFLPQSSLSSEKLFQRSIH
REPGSYAGRRTMQSISNEQKACKVLGIVFFLFVVMWCPFFITNIMAVICKESCNENVIGA
LLNVFVWIGYLSSAVNPLVYTLFNKTYRSAFSRYIQCQYKENRKPLQLILVNTIPTLAYK
SSQLQVGQKKNSQEDAEPTANDCSMVTLGNQHSEEMCTDNIETVNEKVSCV
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| BDBM114603 |
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| n/a |
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| Name | BDBM114603 |
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| Synonyms: | N-[[3-(2-fluorophenyl)-1-methyl-4-pyrazolyl]methyl]-1-[1-(3-methoxyphenyl)-4-pyrazolyl]methanamine | N-[[3-(2-fluorophenyl)-1-methyl-pyrazol-4-yl]methyl]-1-[1-(3-methoxyphenyl)pyrazol-4-yl]methanamine | N-[[3-(2-fluorophenyl)-1-methylpyrazol-4-yl]methyl]-1-[1-(3-methoxyphenyl)pyrazol-4-yl]methanamine | SR-01000757080 | SR-01000757080-2 | [3-(2-fluorophenyl)-1-methyl-pyrazol-4-yl]methyl-[[1-(3-methoxyphenyl)pyrazol-4-yl]methyl]amine | cid_16189988 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H22FN5O |
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| Mol. Mass. | 391.4414 |
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| SMILES | COc1cccc(c1)-n1cc(CNCc2cn(C)nc2-c2ccccc2F)cn1 |
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| Structure | 
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