| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
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| Ligand | BDBM523757 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Binding Assay |
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| Ki | 0.673±n/a nM |
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| Citation |  Witt, KA; Crider, AM; Neumann, W; Hospital, A; Sandoval, K; Kontoyianni, M 3,4,5-trisubstituted-1,2,4-triazoles and 3,4,5-trisubstituted-3-thio-1,2,4-triazoles and uses thereof US Patent US11136312 Publication Date 10/5/2021 |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 4 |
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| Name: | Somatostatin receptor type 4 |
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| Synonyms: | SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 42015.38 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P31391 |
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| Residue: | 388 |
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| Sequence: | MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
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| BDBM523757 |
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| n/a |
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| Name | BDBM523757 |
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| Synonyms: | US11136312, Compound MM-I-87 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H22F4N6 |
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| Mol. Mass. | 482.476 |
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| SMILES | Fc1ccc2c(Cc3nnc(Cc4cccc(c4)C(F)(F)F)n3CCCc3c[nH]cn3)c[nH]c2c1 |
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| Structure | 
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