| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM642197 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Mu-Opioid Receptor Binding Assay |
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| Ki | 18.0±n/a nM |
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| Citation |  Chang, P; Glowaky, R; Rogers, MD Opioid compounds and uses thereof US Patent US11845759 Publication Date 12/19/2023 |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44789.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35372 |
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| Residue: | 400 |
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| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM642197 |
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| n/a |
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| Name | BDBM642197 |
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| Synonyms: | US1184575, 14-acetyl oxycodone |
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| Type | Small organic molecule |
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| Emp. Form. | C20H23NO5 |
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| Mol. Mass. | 357.4003 |
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| SMILES | COc1ccc2CC3N(C)CCC45C(Oc1c24)C(=O)CCC35OC(C)=O |TLB:22:21:16.5.6:8.10.11,THB:15:16:21:8.10.11,9:8:21:16.5.6| |
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| Structure | 
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