| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 52 |
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| Ligand | BDBM652356 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Glosensor cAMP assay |
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| EC50 | 143±33 nM |
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| Citation |  ZHOU, J; ALLEN, JA; WANG, P; FELSING, DE HETEROCYCLIC G-PROTEIN-COUPLED RECEPTOR 52 (GPR52) AGONISTS US Patent US20240059655 Publication Date 2/22/2024 |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 52 |
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| Name: | G-protein coupled receptor 52 |
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| Synonyms: | G-protein coupled receptor 52 | GPR52_MOUSE | Gpr52 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 41353.59 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_117396 |
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| Residue: | 361 |
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| Sequence: | MNESRWTEWRILNMSSSIVNVSEHHSCPLGFGHYSVEDVCIFETVVIVLLTFLIISGNLT
VIFVFHCAPLLHHYTTSYFIQTMAYADLLVGVTCLVPTLSLLHYSTGVHESLTCQVFGYI
ISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIIMIWIYSCLIFLPSFFGW
GKPGYHGDIFEWCATSWLTSAYFTCFIVCLLYAPAALVVCFTYFHIFKICRQHTKEINDR
RARFPSHEVEASREAGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSF
LTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCVCAKDQEAQDPKPRRRANSCS
I
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| BDBM652356 |
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| n/a |
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| Name | BDBM652356 |
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| Synonyms: | US20240059655, Compound PW0864 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H22F3N3O2 |
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| Mol. Mass. | 429.4349 |
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| SMILES | Cc1c(Nc2cc(Cc3ccccc3C(F)(F)F)ccn2)cccc1C(=O)NCCO |
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| Structure | 
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