| Reaction Details |
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 | Report a problem with these data |
| Target | Fatty acid-binding protein 5 |
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| Ligand | BDBM312343 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Time Resolved-Fluorescence Energy Transfer (TR-FRET) Assay |
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| IC50 | 80.0±n/a nM |
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| Citation |  Buettelmann, B; Ceccarelli, SM; Kuehne, H; Kuhn, B; Neidhart, W; Obst Sander, U; Richter, H Bicyclic thiophenylamide compounds US Patent US9604977 Publication Date 3/28/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Fatty acid-binding protein 5 |
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| Name: | Fatty acid-binding protein 5 |
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| Synonyms: | FABP5 | FABP5_HUMAN | Fatty acid binding protein epidermal | Fatty acid-binding protein 5 (FABP5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 15164.79 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q01469 |
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| Residue: | 135 |
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| Sequence: | MATVQQLEGRWRLVDSKGFDEYMKELGVGIALRKMGAMAKPDCIITCDGKNLTIKTESTL
KTTQFSCTLGEKFEETTADGRKTQTVCNFTDGALVQHQEWDGKESTITRKLKDGKLVVEC
VMNNVTCTRIYEKVE
|
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| BDBM312343 |
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| n/a |
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| Name | BDBM312343 |
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| Synonyms: | 2-[3-(4-Trifluoromethyl-thiazol-2-yl)-4,7-dihydro-5H-thieno[2,3-c]pyran-2-ylcarbamoyl]-cyclopent-1-enecarboxylic acid | US9604977, Example 89 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H15F3N2O4S2 |
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| Mol. Mass. | 444.448 |
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| SMILES | OC(=O)C1=C(CCC1)C(=O)Nc1sc2COCCc2c1-c1nc(cs1)C(F)(F)F |t:3| |
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| Structure | 
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