| Reaction Details |
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 | Report a problem with these data |
| Target | Fatty acid-binding protein, adipocyte |
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| Ligand | BDBM312401 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Time Resolved-Fluorescence Energy Transfer (TR-FRET) Assay |
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| IC50 | 10.00±n/a nM |
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| Citation |  Buettelmann, B; Ceccarelli, SM; Kuehne, H; Kuhn, B; Neidhart, W; Obst Sander, U; Richter, H Bicyclic thiophenylamide compounds US Patent US9604977 Publication Date 3/28/2017 |
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| More Info.: | Get all data from this article, Assay Method |
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| Fatty acid-binding protein, adipocyte |
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| Name: | Fatty acid-binding protein, adipocyte |
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| Synonyms: | A-FABP | AFABP | ALBP | Adipocyte lipid-binding protein | FABP4 | FABP4_HUMAN | Fatty acid binding protein adipocyte | Fatty acid-binding protein 4 | Fatty acid-binding protein 4 (FABP4) |
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| Type: | Enzyme |
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| Mol. Mass.: | 14719.23 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P15090 |
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| Residue: | 132 |
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| Sequence: | MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKN
TEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVM
KGVTSTRVYERA
|
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| BDBM312401 |
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| n/a |
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| Name | BDBM312401 |
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| Synonyms: | 2-[6,6-Difluoro-3-(3-trifluoromethyl-[1,2,4]oxadiazol-5-yl)-4,5,6,7-tetrahydro-benzo[b]-thiophen-2-ylcarbamoyl]-cyclopent-1-enecarboxylic acid | US9604977, Example 147 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H14F5N3O4S |
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| Mol. Mass. | 463.378 |
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| SMILES | OC(=O)C1=C(CCC1)C(=O)Nc1sc2CC(F)(F)CCc2c1-c1nc(no1)C(F)(F)F |t:3| |
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| Structure | 
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